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MERTK

MERTK,即MER原癌基因酪氨酸激酶(MerTK),別名PROS1R、TYRO3、Axl-likeprotein等。它是一種受體酪氨酸激酶,屬于TAM(TYRO3、AXL、MERTK)家族成員之一。MERTK在多種組織中表達,包括巨噬細胞和視網膜色素上皮細胞。其作用機制涉及與磷脂酰絲氨酸(PS)暴露的凋亡細胞結合,介導巨噬細胞的吞噬作用,促進細胞凋亡的清除,同時參與調節炎癥反應和免疫應答。MERTK對于維持組織穩態、促進損傷修復、調節免疫反應具有重要作用。MERTK的異常表達與多種疾病相關,包括視網膜色素變性、某些類型的癌癥以及免疫相關疾病。在腫瘤微環境中,MERTK的表達與腫瘤免疫逃逸有關,通過調節腫瘤相關巨噬細胞(TAMs)的吞噬作用,影響腫瘤免疫原性和抗腫瘤免疫。MERTK是癌癥治療中一個潛在的藥物靶點。

熱銷產品

Recombinant Human Tyrosine-protein kinase Mer (MERTK), partial (Active) (CSB-MP621519HU)

驗證數據

CSB-MP621519HU

(Tris-Glycine gel) Discontinuous SDS-PAGE (reduced) with 5% enrichment gel and 15% separation gel.

CSB-MP621519HU

Activity
Measured by its binding ability in a functional ELISA. Immobilized MERTK at 2 μg/ml can bind anti-MERTK antibody(CSB-RA621519A1HU), the EC50 is 32.95-48.25 ng/mL.

CSB-MP621519HU

The purity of MERTK was greater than 95% as determined by SEC-HPLC

MERTK Recombinant Monoclonal Antibody (CSB-RA621519A1HU)

驗證數據

CSB-RA621519A1HU

The Binding Activity of MERTK with anti-MERTK antibody.
Activity: Measured by its binding ability in a functional ELISA. Immobilized MERTK at 2 μg/mL can bind anti-MERTK antibody(CSB-RA621519A1HU), the EC50 is 41.31-72.08 ng/mL.

MERTK Antibodies

MERTK for Homo sapiens (Human)

MERTK Proteins

MERTK Proteins for Rattus norvegicus (Rat)

MERTK Proteins for Homo sapiens (Human)

MERTK Proteins for Mus musculus (Mouse)